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Tamiflu
Antiviral • Neuraminidase inhibitor
Half-life
6-10 hours (active metabolite)
Protein Binding
42%
Metabolized By
Hepatic esterases
External
Drugs.comInhibits influenza neuraminidase, preventing viral release from infected cells
Drug Class
Antiviral
Subclass
Neuraminidase inhibitor
Half-life
6-10 hours (active metabolite)
Time for plasma concentration to decrease by 50%
Protein Binding
42%
Fraction bound to plasma proteins
Therapeutic Index
Wide
Margin between therapeutic and toxic doses