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  3. /Ketorolac

Ketorolac

Toradol, Acular, Omidria, Acuvail, Sprix

NSAID • Pyrrolizine carboxylic acid derivative

Premium
BleedingNephrotoxic

Half-life

5-6 hours

Protein Binding

Metabolized By

CYP2C9

External

Drugs.com

Mechanism of Action

Potent non-selective COX inhibitor with analgesic activity comparable to opioids

Indications(5)

DeQuervain TendinopathyPost Cataract SurgeryPostoperative PainAcute PainOpioid Use Disorder

Classification

Drug Class

NSAID

Subclass

Pyrrolizine carboxylic acid derivative

Brand Names

ToradolAcularOmidriaAcuvailSprix

Key Properties

Half-life

5-6 hours

Time for plasma concentration to decrease by 50%

Protein Binding

—

Fraction bound to plasma proteins

Therapeutic Index

Wide

Margin between therapeutic and toxic doses

Not a substitute for clinical judgement
Ketorolac Drug Profile | PharmaGraphX