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Glucotrol, Glucotrol XL
Antidiabetic • Sulfonylurea
Stimulates insulin release from pancreatic beta cells by closing K-ATP channels
Drug Class
Antidiabetic
Subclass
Sulfonylurea
Half-life
2-4 hours
Time for plasma concentration to decrease by 50%
Protein Binding
98-99%
Fraction bound to plasma proteins
Therapeutic Index
Wide
Margin between therapeutic and toxic doses